Naphthyzinum - instructions for use for children and adults, indications, composition, form of release, dosage and price. Naphthyzine drops - official instructions for use Application of naphthyzine in the nose

Content

According to medical terminology, Naphthyzinum refers to drugs from the group of alpha-adrenergic agonists with a vasoconstrictive effect. Its active substance naphazoline acts on the alpha2-adrenergic receptors of the nasal cavity. The drug is produced by domestic and foreign pharmacological companies. Check out its instructions for use.

Composition of Naphthyzinum

Naphthyzin is available in the form of children's, adult sprays or drops and Naphthyzin Plus. Their composition:

Children's drug

Adult medication

Naphthyzin plus

Description

Clear colorless liquid

Concentration of naphazoline nitrate, %

Auxiliary components

water, boric acid

Boric acid, sea water, sodium hydroxide, water for injection

Package

Glass bottles or dropper bottles of 10, 15, 20 ml in a cardboard box with instructions for use

pharmachologic effect

The drug has a vasoconstrictor effect, pronounced, fast and long-lasting effects. The active component of the composition stimulates alpha-adrenergic receptors, reduces hyperemia, exudation, swelling of the nasal mucosa. With rhinitis, the use of Naphthyzinum facilitates breathing, but after 5-7 days of taking the drops, tolerance (stability) occurs.

Immediately after applying the agent to the mucous membrane, it begins to act locally, providing vasoconstriction. If you use the drug often and for a long time, then naphazoline is partially absorbed, leading to an increase in blood pressure. With intranasal use, the therapeutic effect of the drug occurs after 5 minutes and lasts 4-6 hours.

Why Naphthyzin

All types of the drug have the same indications for use. The instruction identifies the following diseases for which they are effective:

  • acute rhinitis;
  • laryngitis;
  • acute and chronic sinusitis;
  • facilitating rhinoscopy;
  • acute eustachitis;
  • swelling of the larynx due to the development of allergies or radiation therapy;
  • hyperemia of the mucosa after surgery;
  • in ophthalmology: chronic conjunctivitis, asthenopic disorders.

Method of application and dosage

Drops can be used intranasally, instilled into each nasal passage. Adults and children over 15 years old are prescribed 1-3 drops of a 0.1% solution 3-4 times a day. For diagnostic purposes, Naphthyzin is instilled into the nose immediately after cleansing, 3-4 drops, or a swab soaked in a 0.05% solution is injected and left for 1-2 minutes. It can also be used for inhalation. To do this, a 0.05% solution is mixed with saline in equal proportions.

In ophthalmology, it is possible to drip the agent into the eyes as prescribed by the doctor and only after the diagnosis has been established. 1-2 drops of a 0.05% solution are instilled into the conjunctival cavity, the procedure is repeated 1-3 times a day. The first instillation is carried out under the supervision of a doctor, then the patient can independently perform therapy. With stuffy ears, Naphthyzin is also dripped after agreement with the doctor.

Children's Naphthyzinum

A solution with a concentration of naphazoline 0.05% (for children) is not used to treat children under one year old. At the age of 6 years, 1-2 drops are prescribed, 6-15 years old - 2 drops 1-3 times a day. If the vasoconstrictor effect of the child remedy is too strong, the solution is used diluted by half (distilled water is used for dilution), obtaining a 0.025% preparation.

special instructions

In the instructions for use, it is useful to study the special instructions section. Necessary recommendations for patients:

  1. It is forbidden to take the drug simultaneously with monoamine oxidase inhibitors, it is desirable to withstand a break between the use of drugs in 2 weeks.
  2. The use of Naphthyzinum prolongs the effect of local anesthetics used for superficial anesthesia.
  3. Nasal drops are not used for chronic rhinitis.
  4. It is forbidden to take the medicine for more than 5-7 days in a row. This leads to a gradual decrease in the action of vasoconstriction, the manifestation of the effect of tachyphylaxis. Resorptive action and addiction may develop. It is difficult to wean from the use of drops, because gradually the mucous membrane atrophies. Washing, cauterizing blood vessels in the nose, taking certain drugs, or even surgery can help to cope with addiction.
  5. During treatment, it is not forbidden to drive cars or dangerous machinery.
  6. When carrying a child and lactation, Naphthyzinum can be used with caution, weighing the risks for the baby and the benefits for the mother.

Side effects of Naphthyzinum

When using the drug, side effects may develop. The instruction highlights the following:

  • irritation of the mucous membrane;
  • persistent and rapidly developing hyperemia;
  • swelling of the nasal mucosa, atrophic rhinitis - when using the product for more than a week;
  • nausea, vomiting;
  • headache;
  • tachycardia, increased blood pressure - with a predisposition to such phenomena.

When using the drug for a long time or constantly exceeding the dose, the patient's consciousness may be disturbed, blood pressure may increase. For this, the use of Naphthyzin is canceled, symptomatic treatment is prescribed. It is possible to cure addiction and drug overdose by observing individually prescribed therapy. The relief of poisoning in children is carried out only by a doctor.

Contraindications

The use of Naphthyzinum has its own limitations. The instruction highlights the following contraindications:

  • arterial hypertension;
  • hyperthyroidism;
  • intolerance to the ingredients of the composition;
  • atherosclerosis;
  • diabetes;
  • combination with monoamine oxidase inhibitors or a period of less than 14 days from the moment they were discontinued;
  • tachycardia;
  • age up to a year for a 0.05% solution and up to 15 years for a 0.1% solution;
  • serious eye disease.

Terms of sale and storage

You can buy drops without a prescription. The product is stored away from children at a temperature of 10-25 degrees for no longer than three years.

Analogues

You can find an analogue of Naphthyzinum among drugs with the same therapeutic effect or composition, or with a similar effect, but with a different composition. These substitutes include:

  • Nafazolin, Nafazolin-Ferein - nasal drops with a vasoconstrictor effect based on the component of the same name, differ in manufacturer.
  • Naphthyzinum Bufus - drops and spray in the nose for vasoconstriction based on naphazoline.
  • Sanorin - anticongestive and vasoconstrictive nasal drops containing naphazoline nitrate.

Naphthyzinum price

You can buy the drug in pharmacies or via the Internet at a cost that depends on the trade margin and the type of product produced. In Moscow, approximate prices will be:

Medication type

Manufacturer

Internet price, rubles

Pharmacy cost, rubles

Baby drops 0.05%, 10 ml

Dove Pharm, Russia

Update, Russia

Naphthyzinum Renewal drops 0.05% 20 ml

Naphthyzinum Renewal drops 0.1% 20 ml

Adult drops 0.1% 15 ml

Lekko, Russia

Slavyanskaya apteka, Russia

Naphthyzine plus, 0.1%, 15 ml

Groteks, Russia

plus 0.05% 15 ml

Baby drops 0.05% 15 ml

Slavic pharmacy

Adult spray 0.1% 15 ml

Slavic pharmacy

Doctor, Russia

Naphthyzinum - nasal drops to relieve symptoms of nasal congestion. Many use them for years and fall into a real addiction, losing the ability to breathe on their own. Meanwhile, the drug in large doses and with prolonged use is dangerous not only for health, but even for life. Naphthyzinum poisoning in children poses the greatest danger, but overdoses in adults are also not uncommon.

Composition and purpose of Naphthyzinum

The active substance of the anticongestive agent, alpha-adrenergic agonist, or, more simply, vasoconstrictor drops, Naphthyzine is naphazoline. As auxiliary substances, the composition contains purified water and boric acid.

The drug has vasoconstrictive properties, quickly reduces swelling of the nasal mucosa, exudation (discharge), hyperemia (redness).

The use of Naphthyzinum is indicated for:

  • acute catarrhal or allergic rhinitis;
  • sinusitis;
  • eustachitis (inflammation of the auditory tube);
  • to perform the rhinoscopy procedure.

Information about contraindications and side effects

In the annotation to the drug, conditions are prescribed in which Naphthyzin has contraindications for use.

Contraindications

The medicine is contraindicated in:

  • arterial hypertension;
  • tachycardia;
  • diabetes mellitus;
  • severe eye diseases;
  • chronic rhinitis;
  • hyperthyroidism;
  • severe atherosclerosis;
  • hypersensitivity to the components of the drug.

In addition, there are age restrictions for the use of this medication:

  • for a 0.1% solution - up to 18 years;
  • for 0.05% solution - up to 1 year.

Side effects

As a result of prolonged use or the use of high doses of Naphthyzinum, side effects may occur:

  1. Deterioration of the blood supply to the brain and mucous membranes, as a result of which migraine symptoms, nervousness and weakness are observed, in school-age children the ability to learn is reduced, in younger children vision may deteriorate.
  2. Increased blood pressure, headaches.
  3. Swelling and inflammation of the nasal mucosa, hyperemia, dryness, burning in the nose.
  4. Increased heart rate (tachycardia).
  5. Decrease in the duration of action of the drug, provoking the use of higher doses and increase the frequency of their use.

The latter effect is the most common in patients who have used Naphthyzinum for more than 1 week. During this time, the small blood vessels of the nasal cavity adapt to nasal drops, and Naphthyzin ceases to act on them as a vasoconstrictor for a long time. As a result, patients become dependent on the drug, and begin to increase its dosage uncontrollably.

Interaction with alcohol

Due to the fact that the study of the actions of Naphthyzine is still ongoing, and many aspects, including interactions with other drugs and alcohol, are not well understood, it is difficult to talk about the effect of alcohol on the effect of the drug. However, from the experience of practicing physicians, it is known that the intake of alcoholic beverages can cause swelling of the nasal mucosa in patients with dependence on Naphthyzinum, as a result of which they have to "drip" after drinking alcohol.

Is it possible to get poisoned with Naphthyzinum

Given the vasoconstrictive effect of the drug and its ability to be addictive in patients, the question arises whether Naphthyzinum can be poisoned, and how harmful drops are in the treatment of rhinitis in a child.

Consequences of improper treatment

Strictly speaking, Naphthyzinum is not a cure for the common cold as such. These drops serve as an aid to facilitate breathing in various respiratory diseases. Therefore, you can not count on the therapeutic effect of the common cold when using only this drug. And even more so, it is impossible to increase the recommended doses and frequency of Naphthyzinum on your own, because. Is it dangerous.

An uncontrolled increase in doses can lead to dependence on the action of the drug, which will force you to increase its amount even more. And this will already lead to an overdose and poisoning with Naphthyzinum.

Consequences of use in children

Sometimes small children are brought to the intensive care unit, whose parents neglected the warnings in the instructions regarding the age limits for the use of Naphthyzin. The mucous membranes of a small child are much more tender and sensitive than those of an adult. Therefore, even small, according to parents, doses can cause the development of adverse reactions in a child with rather serious consequences. In no case should you use Naphthyzinum, the concentration of which does not correspond to the age of the child or in babies under 1 year old!

What happens if you take the medicine

The worst case scenario can expect a baby who drank the contents of a bottle of Naphthyzinum due to the carelessness of his parents. This happens most often in families with small children, where the mother or other adults are drug dependent on Naphthyzinum. Drops that are used several times a day can be on the couch, under the pillow, on the windowsill, that is, where the baby can easily get them and get drunk.

You can also get poisoned by a low-quality, expired drug, even if you follow all the other rules for use.

Clinical picture in case of overdose and degree of poisoning

Signs of Naphthyzinum poisoning can be manifested by the following symptoms:

  • abdominal pain, nausea;
  • slow heart rate (bradycardia);
  • lowering blood pressure;
  • dizziness, drowsiness, lethargy, in children - a sharp deterioration in mood;
  • appearance of cold sweat on the skin, blanching.

These symptoms can be both mild and pronounced. The clinical picture depends on the degree of overdose.

  • A mild degree of intoxication is manifested by one or more symptoms that quickly disappear when the drug is discontinued and do not require medical intervention.
  • The average degree is usually detected by several symptoms at once, but when you stop using Naphthyzin, it goes away on its own and also does not require the patient to be hospitalized.
  • A severe degree is the most dangerous, since it primarily disrupts the heart rate - from tachycardia to bradycardia, vomiting and other signs of intoxication may occur, and if measures are not taken, a person may fall into a coma.

Of course, at the first suspicion of a severe degree of Naphthyzinum poisoning, it is necessary to call an ambulance.

How to provide first aid to the victim

The danger of poisoning lies in the fact that the longer the victim is not helped, the more widespread intoxication in the body. The consequences of extensive intoxication can be difficult to predict and sometimes the patient cannot be saved. In order to alleviate the condition of the poisoned person and prevent the further spread of intoxication, it is worth being vigilant before the arrival of doctors.

  • Be careful to keep the victim conscious.
  • Constantly monitor his respiratory function and heart rhythms.
  • Put the victim to bed, cover with a warm blanket and let's drink plenty of warm drinks.
  • Watching the pulse, remember or write down its changes, the information may be needed by doctors.

Treatment in a hospital

When the victim is admitted to the hospital, blood will first be taken for biochemical analysis and an electrocardiogram will be made.

  1. If the poisoning occurred as a result of an overdose during use, then most often the treatment consists in taking sorbents (for example, Enterosgel).
  2. If Naphthyzin was drunk, be sure to wash the stomach, prescribe sorbents and symptomatic therapy.
  3. If bradycardia is detected, a subcutaneous injection of an antidote, atropine sulfate, is made.
  4. In severe cases, the introduction of Prednisolone may be required, in extremely severe cases, Dopamine, infusion therapy is used.
  5. With the moderate severity of Naphthyzinum poisoning, the use of rehydrating solutions is effective. As a rule, in 30-60 minutes, all manifestations of intoxication can be stopped.

The cheapness and availability of the drug provokes people with chronic forms of rhinitis to use the drug uncontrollably and treat their children on their own. But the consequences of an overdose can bring incomparably large expenses for saving the victim from poisoning, not to mention the damage to the health of the poisoned person. Therefore, the use of Naphthyzinum is recommended for 5-7 days, no more.

If after this time the nasal congestion does not go away, you should look for the causes of a prolonged runny nose and other methods of treatment. And for those who are already firmly “addicted” to Naphthyzin, we can advise you to quit it in one motion, in the morning. The first time will be difficult, but no more than 2-3 days. Then the respiratory function will be restored, and you will feel complete freedom from not very useful drops.

December 9, 2015

The use of Naphthyzinum should not last longer than a week, because as a result, patients may experience side effects. With long-term treatment with a solution, patients may no longer feel relief from the action of naphazoline.

If the patient is taking monoamine oxidase inhibitors (nialamide or befol), then the attending physician should be warned about this. Such drugs should not be combined with the treatment of the common cold with Naphthyzinum. Even after stopping taking MAO inhibitors, you must wait 10 days, and then start treating rhinitis with a vasoconstrictor.

Side effects

At the first injection of the Naphthyzine solution in any percentage, patients may experience severe dryness in the nose, a slight burning sensation or a feeling of tightening of the tissues. But in a short time, these negative manifestations disappear, and the patient ceases to feel discomfort in the nasal cavity.

With prolonged use, Naphthyzin may lose its positive effects. If this is noted, then the patient needs to stop the introduction of a vasoconstrictor solution. Exceeding the duration of treatment can lead to some degenerative changes in the membrane of the nasopharynx.

Contraindications

As well as preparations containing chemical elements, Naphthyzin is contraindicated in certain diseases. The drug is prohibited for use in patients with the following pathologies:

  • Cardiopalmus
  • Tendency to increase pressure
  • hyperthyroidism
  • Atherosclerosis
  • Children up to a year
  • Individual sensitivity to components

Before the introduction of Naphthyzinum, it is imperative to consult a therapist so as not to harm health.

Overdose symptoms

With prolonged treatment with Naphthyzinum, the patient may experience negative reactions of the body. Exceeding the dosage of the drug indicated by the ENT can cause serious complications, such as increased pressure and dizziness. This is due to the fact that at high doses, a solution of naphazoline penetrates into the blood and has a resorptive effect.

If the patient has symptoms of an overdose, it is necessary to stop treatment with Naphthyzinum and contact an ENT. Sympatholytic therapy may be required to eliminate negative effects.

Interaction with drugs

Naphthyzinum is not recommended to be used simultaneously with drugs aimed at lowering blood pressure. If it is still necessary to administer a nasal remedy and drink antihypertensive tablets, then Naphthyzinum is used with extreme caution. And in cases where the treatment of hypertension is more important for the patient, it is better to abandon the vasoconstrictor solution altogether.

CNS stimulant drugs will enhance the effects of naphazoline.

Naphthyzin for children: features

The adult dosage of Naphthyzinum is not used in the treatment of rhinitis in children under five years of age. At this age, in babies, naphazoline can affect the nervous system, causing negative developmental consequences and reactions. A vasoconstrictor can depress the child's central nervous system. And children 6-12 years old can be administered Naphthyzin only once a day.

If the child has repeated bleeding from the nose, then swabs soaked in Naphthyzine 0.05% solution can be used to stop. This drug has a vasoconstrictive and hemostatic effect.

Children's Naphthyzinum is used in the treatment of rhinitis in babies from the first year of life. Newborns are not recommended to inject naphazoline into the nasopharynx.

  • A child from a year old is prescribed Naphthyzinum 0.025%. During the day, you can drip 1-2 drops into each nasal passage. Repeat the procedure twice a day.
  • Naphthyzine 0.05% is also used in the treatment of childhood rhinitis. Based on age, the ENT should prescribe the exact dosage and frequency of instillation.

Unlike the adult concentration of the drug, the children's decongestant contains a minimal amount of the active ingredient. It is prescribed for acute inflammation of the nasopharynx and during nosebleeds.

How is Naphthyzin used in pediatrics?

The active ingredient in children's Naphthyzinum is naphazoline, which has the form of a coarse yellow powder. It practically does not interact with water, but is perfectly diluted with alcohol. The drug relieves the inflammatory process, reduces swelling of soft tissues and eliminates rhinorrhea. During a runny nose in children, Naphthyzin reduces blood flow to the blood vessels, thereby providing good ventilation in the nasal cavity.

In pediatrics, the drug is used for acute rhinitis, sinusitis, bleeding. But, since Naphthyzinum can cause serious side effects, it is not used as often in the treatment of ENT diseases as other safe drugs.

Especially avoid the use of naphazoline for the treatment of infants. It is very difficult for babies to measure the exact dose of the solution, which will not cause overdose symptoms. But children from a year are prescribed Naphthyzin 0.025%. A child from 5 years old can already increase the concentration of the active substance and administer the drug 0.05%.

But even when using low concentrations of naphazoline, children should not overdose on a vasoconstrictor. The maximum number of drops is 2 in each nostril. The duration of treatment should not exceed 5 days. If the child needs a longer period of use of the decongestant, then only the doctor can make this decision.

When children are concerned about frequent nosebleeds, a 0.05% solution of Naphthyzinum is used to stop them. A cotton flagellum is impregnated with a medicinal liquid and injected into the nostril, from which blood flows. You need to hold it for a couple of minutes, and then you can take it out.

How not to overdose children's Naphthyzinum?

Since the vasoconstrictor active component of the drug naphazoline is a selective adrenomimetic, it acts almost like adrenaline. Although it is a very effective topical remedy for the common cold, it can cause tachyflaxia. That is, the body of a child or an adult patient after a short period of use of Naphthyzinum begins to get used to the action of alpha-agonists and stops responding to the drug.

As a result, patients in the nasal cavity begin to develop drug-induced rhinitis. Children are especially susceptible to tachyflaxia, because the risk of overdosing the solution is much higher than in adults. In addition, often the patients themselves contribute to the fact that they develop dependence on Naphthyzinum. This happens in cases where the agent ceases to effectively act on the nasal mucosa and, in order to increase the ability of the drug to relieve swelling, parents increase the dose of naphazoline solution or instill drops more often than the period indicated in the instructions.

Recall that the maximum time of application of Naphthyzinum is 5-7 days. Further, if you need to increase the duration of treatment, you need to consult a doctor or replace one drug with a more effective and safe one. In some cases, the ENT recommends stopping the introduction of naphazoline into the nasal cavity, taking a break for several days, and then using a medicine from another group of vasoconstrictor drugs.

According to the instructions, Naphthyzinum in a children's dosage should not be instilled in newborns and infants up to a year. And only a specialist can prescribe this medicine to a child from 1 year of age, after he has assessed all the risks and calculated a safe dosage.

If Naphthyzin was attributed to children from a year old, then parents should know one nuance. The factory plastic packaging does not contain an accurate dropper, so it is very easy to overdose the medicine. In order to avoid introducing a larger amount of solution into the baby's nose, it is better to take an ordinary pipette and bury Naphthyzin drop by drop, without fear of an overdose and drug poisoning.

Another point that you need to pay attention to is the observance of the frequency of instillation of the nasal cavity in children. The instructions say that the procedure can be repeated up to 4 times a day. If the puffiness does not subside or the effect is not felt as much as we would like, it is not necessary to increase the frequency of instillation of the spout. Experts advise additionally rinsing the nasopharynx with saline solutions, for example, Aquamaris or using Pinosol oil drops.

Naphthyzine 0.1% should not be used for the treatment of children's rhinitis. If there is no other option, then the agent is diluted with distilled water (1: 1). But this can be done only as a last resort.

Naphthyzinum can be used in the treatment of the following pathologies:

  • Acute rhinitis of any origin
  • Syringitis
  • Laryngitis
  • Swelling of the nasopharynx, larynx
  • Conjunctivitis of a bacterial nature

But, if the child has arterial hypertension, atherosclerosis or diabetes mellitus, then Naphthyzin is forbidden to use. Also, do not administer the solution for chronic rhinitis and hyperthyroidism.

When a baby accidentally drinks a vasoconstrictor, he may experience serious symptoms: pressure drop, drowsiness, collapse. The action of naphazoline resembles Clonidine, which depresses the central nervous system and provokes a decrease in blood pressure to a minimum. As soon as the parents see the symptoms of an overdose of Naphthyzinum, it is necessary to call an ambulance. At home, you need to quickly rinse the stomach with warm water and give activated charcoal tablets per 1 pc. for every 10 kg of the child's weight.

If the nose is stuffy and it becomes very difficult to breathe, expectant mothers go to the pharmacy for some effective medicine. Can Naphthyzinum be used during pregnancy?

In order to answer this question, you need to refer to the instructions. It states that although the drug is not strictly prohibited, it can still be used only in situations where there is no other way to get rid of rhinitis. If the doctor prescribes Naphthyzinum during pregnancy, then the woman should strictly monitor compliance with dosages and not exceed the daily frequency of administration of the solution into the nasal cavity.

Runny nose in pregnant women appears quite often. During this period, a woman becomes especially vulnerable to various colds, as well as the progression or appearance of allergic rhinitis. Even if the expectant mother does not have SARS or allergies, she may experience the so-called "pregnant runny nose", which is caused by changes in the hormonal background. If the nose is blocked for this reason, then it makes no sense to use Naphthyzin and is even prohibited.

Sometimes a vasoconstrictor drug is prescribed to pregnant women when drugs from another group have been tried, but they have not shown proper results in the treatment of the common cold. Tolerating nasal congestion and not being able to fully breathe is also prohibited, because a lack of oxygen can lead to fetal hypoxia. But taking a vasoconstrictor can also narrow the tissues and blood vessels of the placenta, blocking the access of air to the child being born. Obviously, the risk is quite high, so a pregnant woman should in no case self-medicate using Naphthyzin without a doctor's recommendation.

When a specialist decides to prescribe a nasal drug with naphazoline, then he must carefully calculate the dosage of the drug. It is also important not to use vasoconstrictor chemicals during the 1st trimester of pregnancy.

It is not recommended to inject Naphthyzin into the nasal cavity for more than 3 days, because a woman may become addicted to the active ingredient. It is best to use the drops at bedtime so that mom can sleep well at night. During the day, you can replace Naphthyzinum with other, safer sea salt solutions or saline solutions. Inhalations, acupressures of the nose also help well. These methods of treating a runny nose will not be addictive and will not cause developmental disorders in the baby.

Is it possible to use children's Naphthyzinum during pregnancy?

In some cases, pregnant women believe that if the drug is available in a children's dosage and is safer than drugs for adults, then it may well be used in the treatment of their common cold. But this is far from true.

Children's Naphthyzinum 0.05% is prescribed for babies in extreme cases, when it is not possible to eliminate the swelling of the nose with any other medicines. The concentration of the active ingredient is relatively lower, but this does not mean that it becomes harmless. It really has a lesser negative effect on the patient's body, but it can still harm a pregnant woman and her fetus.

Naphthyzine with a low concentration of 0.025% naphazoline should not be taken as a completely safe vasoconstrictor. That is, the drug is not prohibited for use by pregnant women, but its use is undesirable.

The exact contraindications to the use of Naphthyzinum during pregnancy are the following diseases or abnormalities:

  • High blood pressure and heart palpitations
  • Severe atherosclerosis
  • Chronic runny nose
  • High sensitivity to the active substance

The attending physician who will prescribe Naphthyzinum will first exclude serious diseases that adrenomimetics can have a negative impact on and, only after that, will recommend the dosage of the drug.

What to do if you develop dependence on Naphthyzinum?

One of the first side effects that develop after prolonged or frequent administration of naphazoline into the nasal cavity is mucosal addiction. As a result, the shell stops responding to drops of Naphthyzinum and there is no improvement in the condition.

Dependence on naphazoline develops as follows: the period of effective action of the substance decreases, so the patient increases the dose of the drug in order to get quick relief. Constant exposure to Naphthyzinum negatively affects mucous tissues. The patient's sense of smell decreases, dryness appears, crusts constantly form.

Since the functions of the mucosa are inhibited, blood circulation also becomes less active. Due to this, an insufficient amount of blood with nutrients enters the patient's brain, so the patient feels constant fatigue, incapacity to work, and becomes irritable.

As soon as the patient notes such a negative moment, he should immediately stop treatment with a vasoconstrictor drug. A break between therapy (at least 7 days) will be able to restore the normal functionality of the nasal mucosa. But it is important to remember that adrenomimetics themselves provoke a loss of vascular tone over time, which is why they lose the ability to narrow and reduce swelling of tissues.

If the patient has already developed dependence on Naphthyzinum, it is not easy to deal with such a problem. With a sharp cessation of the drug, the patient may experience severe swelling of the mucous membrane and a runny nose will begin again. Chronic rhinitis must be treated.

To do this, you should contact a specialist who can make an accurate diagnosis and prescribe effective remedies to eliminate complex symptoms. First of all, a person needs to stop the uncontrolled use of any nasal preparations, whether it be a spray or drops containing naphazoline. At first, it will be very difficult to get rid of a runny nose, but over time, the mucous membrane will recover and lasting relief will come.

With a strongly neglected mucosal addiction, when the tissue began to grow and breathing through the nose is almost completely blocked, it may be necessary to eliminate the problem surgically. Such operations are performed under local anesthesia and are not accompanied by large blood loss. The specialist uses radio wave technology to reduce the volume of the mucous membrane. After the procedure, the vascular tissue is scarred, and nasal breathing becomes full very quickly.

How to avoid drug rhinitis?

All vasoconstrictor drugs containing adrenergic agonists can cause drug-induced rhinitis. In order to prevent the pathological growth of the vascular network in the mucous membrane, drugs containing active components from the group of alpha-adrenergic agonists should not be used uncontrollably. These include Naphthyzinum, Sanorin, Nazol, Phenylephrine and the like.

The first rule of safe use of vasoconstrictor drugs is to limit the administration of the solution to 4 days in a row. Before use, you need to study the instructions well and strictly adhere to the dosage. If you are not sure that the remedy is suitable, you should definitely consult with an ENT.

It is important to know that Naphthyzinum is not a nasal drug that treats rhinitis of any etiology. It contains components that can only remove puffiness, but not eliminate the cause of inflammation. Accordingly, Naphthyzin only temporarily eliminates the symptoms of the disease, and complex therapy will be required for a complete recovery.

The solution for instillation into the nose refers to alpha-adrenergic agonists, which in most cases are used in ENT practice. What are Naphthyzin drops used for?

The medicine is made in the form of a solution for instillation into the nasal cavity. Available without a prescription in regular vials or dropper bottles of 10 milliliters.

The structure of the drug

The composition of drops "Naphthyzin" includes one active ingredient - naphazoline. Depending on its content in solution, the drug is produced in 0.1% and 0.05%.

Pharmacological properties

The solution belongs to the group of alpha-agonists and has a pronounced narrowing effect on the capillaries. When the drug is instilled into the nasal passages, the pharmacological effect develops after a few minutes and lasts up to four to six hours.

When the medication enters the mucous areas of the nose, the severity of edema and redness decreases, the amount of discharge from the nasal passages decreases significantly.

Indications

According to the instructions for use, Naphthyzin nose drops are prescribed to patients when they have the following conditions and ailments:

  • Acute rhinitis (inflammation in the nasal mucosa).
  • Eustachitis (inflammatory lesion of the auditory tube, leading to a deterioration in the ventilation of the tympanic cavity with the development of catarrhal otitis media).
  • Otitis media (an infectious inflammatory process characterized by rapid development and localized in the middle ear).
  • Bleeding from the nose.
  • Allergic rhinitis (a disease that develops as a result of contact of allergens with the nasal mucosa).
  • Laryngitis (inflammation of the mucous membranes of the larynx, which is associated with colds or infectious diseases such as scarlet fever and whooping cough).
  • (inflammatory disease of the nasopharynx of an infectious-allergic nature).
  • Chronic conjunctivitis (a long-term inflammatory process in the mucous region of the eye, which is characterized by moderate swelling of the eyelids, as well as photophobia, increased tearing).
  • Asthenopia (visual impairment, which is accompanied by increased fatigue in the implementation of visual work).
  • Sinusitis (inflammatory lesion of the mucous membrane of the paranasal sinuses).

Restrictions

Before starting treatment with a medicine, it is necessary to familiarize yourself with the annotation, since the solution has a number of specific contraindications. According to the instructions for use, Naphthyzin drops are forbidden to be used for the following diseases and conditions:

  • Increased blood pressure.
  • Angle-closure glaucoma (a pathological process that leads to injury to the optic nerve).
  • Individual intolerance to the drug.
  • Pregnancy.
  • Lactation.
  • The age of the patient is up to one year and six years (depending on the content of the active ingredient).
  • Hyperthyroidism (a disease that is caused by an increase in the hormonal activity of the endocrine system and is characterized by excessive production of thyroid hormones).
  • Atherosclerosis (a chronic disease of the arteries resulting from a violation of lipid metabolism and accompanied by the deposition of cholesterol in the capillaries).
  • Chronic inflammation of the nasal mucosa.
  • Tachycardia (a sharp increase in heart rate, a sign of serious disorders).
  • Heart rhythm disturbances.
  • Diabetes mellitus (a chronic metabolic disorder, which is based on a lack of production of one's own insulin and an increase in blood sugar levels).

Instruction

What are Naphthyzin drops for? The solution is used intranasally. The dosage regimen is prescribed by the doctor depending on the indications.

To improve nasal breathing and eliminate swelling of the nasal mucosa, the medication is instilled one or two drops into each nostril, tilting your head to the side.

According to the instructions, Naphthyzin nasal drops should not be used for more than five days. In the absence of a positive pharmacological effect, the therapy is stopped and the medical specialist is re-addressed to clarify the diagnosis and select another drug.

For diagnostic studies - after cleansing the nasal passages, you need to drip three to four drops or insert a cotton swab dipped in a 0.05% solution and leave for one to two minutes.

What are Naphthyzin drops for? In case of swelling of the vocal cords, apply 2 milliliters of the solution in the form of a spray (dropper bottle) or in small doses with a special syringe. For bleeding, swabs moistened with 0.05% of the drug are used.

In ophthalmology, "Naphthyzin" is used, one or two drops of a 0.05% solution into the conjunctival cavity and the back surface of the eyelids (three times a day). As an additional agent for superficial anesthesia - four drops per 1 milliliter of local anesthetic.

From what age can you use

The instruction to the drug prohibits the treatment of children under the age of one year with Naphthyzinum. A child from one year old is allowed to use the medication, but many pediatricians prefer to treat rhinitis with drugs based on xylometazoline or oxymetazoline.

According to the instructions for Naphthyzinum, it is forbidden for children to drip nose drops even at a minimum concentration (0.05%) without the doctor's permission. A drug with a concentration of 0.1% is usually not prescribed to small patients, since it is contraindicated under the age of eighteen years.

At the age of one to fifteen years, only 0.05% Naphthyzin is used in such a single dosage:

  1. For children from one to six years - one drop.
  2. For children from six to fifteen years - two drops.

So much of the drug is injected first into one nostril, laying the baby on a flat surface and slightly turning his head so that the medicine hits the wall of the nasal passage. In the future, the procedure is repeated for the second nostril. The frequency of use of the drug is from one to three times a day.

But even with the use of small dosages of the drug, it is not recommended to use a vasoconstrictor drug in high dosages in the treatment of children. The maximum number of drops is two in each nasal passage. The duration of therapy should not exceed five days. If the baby needs a longer course of treatment in the future, then only the doctor can decide which drug to use.

Why are Naphthyzin drops still used? When young patients are concerned about regular nosebleeds, a 0.05% solution is used to neutralize them. A cotton pad is soaked with medicine and injected into the nostril. You need to keep it for a couple of minutes, and then you can remove it.

Use during pregnancy

The safety of Naphthyzinum for women during pregnancy and intrauterine development of the fetus has not been confirmed, therefore this drug cannot be used during this period of time.

Treatment with this medication is carried out only in the presence of serious diseases in a situation where the expected benefit outweighs the risk to the unborn baby. For women during pregnancy, it is best to use the drug in a child dosage. Therapy should be continued no longer than three days.

If you need to use the medication during lactation, you should consult a doctor. It may be best to stop breastfeeding while treatment is in progress.

Negative Effects

According to the instructions, Naphthyzin drops can provoke the appearance of some negative reactions:

  • Burning in the nasal cavity.
  • Stinging in the nasal passages.
  • Constant sneezing.
  • Feeling of dryness in the nose.
  • Migraine (a neurological disease characterized by periodic or regular attacks of pain on one side of the head).
  • Increased fragility of capillaries.
  • Drowsiness.
  • Lethargy.
  • Hyperemia of the nasal mucosa (blood overflow of the vessels of the circulatory system of any organ or area of ​​the body).
  • Edema.
  • Urticaria (a disease of an allergic nature, which is manifested by the formation of blisters on the surface of the skin and on the mucous membranes).
  • Quincke's edema (a disease that is characterized by the appearance of a clearly limited angioedema of the skin, as well as subcutaneous tissue).

Overdose

If the drug is used too often (more than 3-4 times a day) and if more than 2 drops are instilled into the nasal passage, a person may develop symptoms of poisoning, which are expressed in an increase in the above negative effects, as well as weakness, dizziness, palpitations, increased levels blood pressure.

If such phenomena occur, drug treatment should be stopped and a medical specialist should be consulted for complex therapy.

Is it possible to use Naphthyzin with other drugs

The solution, when used together with drugs from the group of local anesthetics, slows down and reduces their pharmacological action.

According to the instructions for use for Naphthyzin drops, it is known that it is not recommended to use it simultaneously with antidepressants. If a person has used drugs of this group, then at least fourteen days must pass before starting therapy with a solution.

It is not recommended to use the drug for more than seven days, because in this case the patient becomes addicted to the active substance, which requires the use of ever larger dosages. Accordingly, the risk of negative phenomena and symptoms of poisoning increases.

If during therapy with this medication a person develops drowsiness or lethargy, then the use of the solution is immediately canceled and the doctor is consulted.

Analogues

In pharmacies, you can find drugs that are similar in their pharmacological effect to Naphthyzinum.

Such medicines include:

  1. "Pharmazolin".
  2. "Xymelin".
  3. "Galazolin".
  4. "Afrin".
  5. "Sanorin".
  6. Aqua Maris.
  7. "Otrivin".
  8. "Rinostop".
  9. Nazivin.
  10. "Tizin".
  11. "Knoxprey".

Before replacing the drug, the patient should consult with a medical specialist about the dosage, prohibitions on the use and duration of the course.

Holiday conditions

Drops "Naphthyzin" can be bought at a pharmacy without a doctor's prescription. Keep the vial of the drug away from children. Storage temperature - no higher than twenty-five degrees.

An open vial should be used within a month. If the medication has not been used, it is disposed of. The shelf life of the medicine in a closed package is twenty-four months. At the end of this time, the product must be thrown away. The cost of the drug varies from 130 to 160 rubles.

Patients' opinions about the drug

There are various reviews about "Naftizin". Patients call this drug both emergency medical care for a runny nose and other diseases, and a drug that provokes addiction. Patients note that this drug can be used for severe symptoms, but it should not be used longer than the time recommended by the doctor.

On the treatment of young patients "Nafthyzinum" respond differently. The drug is called affordable and inexpensive, so it is often used for rhinitis in children. According to the parents, the drug acts effectively and instantly helps to eliminate signs of inflammation for about six hours.

But such a short exposure is also attributed to the negative aspects of the drug. Because of this, most mothers often prefer other vasoconstrictor medications that eliminate nasal congestion for a longer time. In addition, in many responses, patients complain about dependence on Naphthyzinum, which is manifested by a decrease in the effectiveness of the drug.

In cold weather, many people suffer from a runny nose. With a stuffy nose, it is difficult to lead a normal life. There are many remedies for the common cold, but there are inexpensive drops of Naphthyzinum that will help you breathe freely almost immediately after their use. What is the composition of this drug and how to use it correctly for children?

Naphthyzine properties: composition

This remedy for the common cold is one of the most popular medicines. This inexpensive and affordable tool has been used for a long time. At the first sign of nasal congestion, vasoconstrictors are usually used.

These drops have such an effect, and besides, they are considered safe. Is this really so and how to use it correctly to treat the common cold in children and adults?

To understand how safe and effective it is, you need to know the composition of the product. The main component in Naphthyzinum is naphazoline nitrate. This substance is included in the group of alpha - andrenostimulators. The tool also contains the following components:

  • boric acid;
  • prepared (purified) water.

Boric acid has antipruritic and antiseptic action. Naphthyzine is able to actively and effectively remove swelling and redness of the mucosa, reduce the amount of blood passing through the capillaries in the nose and reduce the secretion of mucus.

Such properties of nasal drops allow them to be used in the treatment of many diseases:

  • Rhinitis.
  • Sinusitis.
  • Sinusitis.
  • Allergic rhinitis.
  • Condition after surgery.

Naphthyzinum drops are released into the nose with different concentrations - 0.1% and 0.5% naphazaline nitrate. For the treatment of children, drops with a lower concentration are used. The release form can be nasal drops and spray. It is a clear, colorless solution or slightly colored.

Drops after application act very quickly, so the patient experiences relief almost immediately, can breathe freely.

It should be noted that such an effect is short-term and if you do not use special medicines for the common cold, the dose of Naphthyzinum each time will have to increase.

With the constant use of these drops, drug dependency, as well as atrophy of the vessels of the nasal mucosa, and other diseases. It is very difficult to get rid of such conditions later.

Most patients buy Naphthyzin on their own without a doctor's prescription and start dripping them with nasal congestion. You can always buy such drops in a pharmacy, especially since they cost a penny. However, such a remedy without proper application bad for health which the patient is unaware of.

It is necessary to stop using it for a few days so that the vessels are weaned from the remedy. In more complex forms of addiction, surgery is required. To prevent such conditions, it is necessary to use Naphthyzin according to instructions by application.

When used correctly, the mucosal vessels are reduced. The secretion of mucus becomes much less or stops completely. The ventilation of the paranasal sinuses is normalized, as a result of which nasal breathing becomes quite normal.

Naphthyzin: instructions for use

Nasal drops and spray Naphthyzin are applied topically. Adult patients are recommended to enter into each nasal cavity 1-3 drops of 0.1% solution. The procedure should be carried out 3-4 times a day, trying to adhere to the same time interval.

Naphthyzin drops 0.5% are also used to stop nosebleeds. For this, a cotton swab is moistened in a solution of nasal drops and injected into the nasal passages.

Regardless of the age of the patient, the course of treatment according to the instructions should not exceed 5-7 days. If you continue to apply the drops further, then they will lead to psychological dependence, and medical rhinitis will also begin to develop.

Children's Naphthyzinum is produced with the lowest concentration of the main substance of 0.05% solution. Pediatricians are allowed to use such a drug for children after 1 year of life. Adults also often use it for nasal congestion.

It is recommended for babies to drip 1-2 drops every 6-8 hours. Pediatricians recommend using it for severe nasal congestion with great swelling and mucus secretion. Before using the medicine, it is necessary to clean the nose of the child and only then carefully drip the nose, strictly observing the dosage.

In recent years, cases of exceeding the dosage of Naphthyzinum have become more frequent, and for this reason, many children were poisoned at the age of 1 to 3 years. For children, it is allowed to use children's Naphthyzinum no more than three days.

During this period, it is usually possible to eliminate nasal congestion and the child can breathe freely. If the condition does not improve significantly, lavage of the nasal passages is usually performed.

Side effects of Naphthyzinum

With prolonged use of Naphthyzinum in adults and children, excessive mucosal edema begins. In addition, other side effects also appear:

If you use such a medication for a long time, an addiction appears, from which it is then difficult to get rid of. The body gets used to it and the drops no longer show their effectiveness, but only harm health. In children under 1 year after the use of the nasal preparation, not only mucosal edema begins, but also body poisoning.

It is accompanied by the following symptoms:

  1. Refusal to eat.
  2. Drowsiness.
  3. Indifference.
  4. Low pressure.
  5. Bradycardia.
  6. In some cases, a decrease in body temperature.

With the use of these drops, up to 1 year old, the child's blood pressure and heart rate decrease to the lower limit. Skin turns pale, becomes cold and a child in this state may be in a coma.

Such a remedy for the common cold has many side effects, therefore, if used improperly, it is harmful to the health of adults and especially children. Pediatricians rarely prescribed children's Naphthyzin to small patients, replacing them with more natural and harmless drugs for the child's body.

Naphthyzinum: contraindications

These drops in any concentration have contraindications, these include the following:

Pediatricians always prescribe children's Naphthyzinum with caution to children aged 1 to 6 years. Do not take Naphthyzinum pregnant women and lactating mothers.

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